H(1)-receptor antagonist (CHEBI:37955)

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CHEBI:37955 - H₁-receptor antagonist

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ChEBI Name	H₁-receptor antagonist

ChEBI ID	CHEBI:37955

ChEBI ASCII Name	H1-receptor antagonist

Definition	H₁-receptor antagonists are the drugs that selectively bind to but do not activate histamine H₁ receptors, thereby blocking the actions of endogenous histamine.

Stars	This entity has been manually annotated by the ChEBI Team.

ChEBI Ontology
Outgoing	H₁-receptor antagonist (CHEBI:37955) is a histamine antagonist (CHEBI:37956)

Incoming	(S)-carbinoxamine maleate (CHEBI:59330) has role H₁-receptor antagonist (CHEBI:37955) N-demethylmirtazapine (CHEBI:143428) has role H₁-receptor antagonist (CHEBI:37955) acrivastine (CHEBI:83168) has role H₁-receptor antagonist (CHEBI:37955) alcaftadine (CHEBI:71023) has role H₁-receptor antagonist (CHEBI:37955) antazoline (CHEBI:84115) has role H₁-receptor antagonist (CHEBI:37955) aripiprazole (CHEBI:31236) has role H₁-receptor antagonist (CHEBI:37955) aripiprazole lauroxil (CHEBI:90930) has role H₁-receptor antagonist (CHEBI:37955) astemizole (CHEBI:2896) has role H₁-receptor antagonist (CHEBI:37955) azatadine (CHEBI:2946) has role H₁-receptor antagonist (CHEBI:37955) azatadine maleate (CHEBI:2947) has role H₁-receptor antagonist (CHEBI:37955) azelastine (CHEBI:2950) has role H₁-receptor antagonist (CHEBI:37955) azelastine hydrochloride (CHEBI:2951) has role H₁-receptor antagonist (CHEBI:37955) benzquinamide (CHEBI:27662) has role H₁-receptor antagonist (CHEBI:37955) benzylpenicillin clemizole (CHEBI:52139) has role H₁-receptor antagonist (CHEBI:37955) bepotastine (CHEBI:71204) has role H₁-receptor antagonist (CHEBI:37955) bepotastine besylate (CHEBI:31281) has role H₁-receptor antagonist (CHEBI:37955) bromazine (CHEBI:59177) has role H₁-receptor antagonist (CHEBI:37955) bromazine hydrochloride (CHEBI:59178) has role H₁-receptor antagonist (CHEBI:37955) brompheniramine (CHEBI:3183) has role H₁-receptor antagonist (CHEBI:37955) carbinoxamine (CHEBI:3398) has role H₁-receptor antagonist (CHEBI:37955) carbinoxamine maleate (CHEBI:31353) has role H₁-receptor antagonist (CHEBI:37955) cetirizine (CHEBI:3561) has role H₁-receptor antagonist (CHEBI:37955) chlorphenamine (CHEBI:52010) has role H₁-receptor antagonist (CHEBI:37955) cinnarizine (CHEBI:31403) has role H₁-receptor antagonist (CHEBI:37955) clemastine (CHEBI:3738) has role H₁-receptor antagonist (CHEBI:37955) clemastine fumarate (CHEBI:3739) has role H₁-receptor antagonist (CHEBI:37955) clopenthixol (CHEBI:59115) has role H₁-receptor antagonist (CHEBI:37955) cyclizine (CHEBI:3994) has role H₁-receptor antagonist (CHEBI:37955) cyclizine hydrochloride (CHEBI:51045) has role H₁-receptor antagonist (CHEBI:37955) cyproheptadine (CHEBI:4046) has role H₁-receptor antagonist (CHEBI:37955) cyproheptadine hydrochloride sesquihydrate (CHEBI:650917) has role H₁-receptor antagonist (CHEBI:37955) deptropine (CHEBI:50189) has role H₁-receptor antagonist (CHEBI:37955) deptropine citrate (CHEBI:50190) has role H₁-receptor antagonist (CHEBI:37955) desipramine (CHEBI:47781) has role H₁-receptor antagonist (CHEBI:37955) desloratadine (CHEBI:291342) has role H₁-receptor antagonist (CHEBI:37955) dexbrompheniramine (CHEBI:59269) has role H₁-receptor antagonist (CHEBI:37955) dexbrompheniramine maleate (CHEBI:59273) has role H₁-receptor antagonist (CHEBI:37955) dimenhydrinate (CHEBI:4604) has role H₁-receptor antagonist (CHEBI:37955) diphenhydramine (CHEBI:4636) has role H₁-receptor antagonist (CHEBI:37955) diphenhydramine hydrochloride (CHEBI:4637) has role H₁-receptor antagonist (CHEBI:37955) diphenhydramine salicylate (CHEBI:34720) has role H₁-receptor antagonist (CHEBI:37955) diphenylpyraline (CHEBI:59788) has role H₁-receptor antagonist (CHEBI:37955) diphenylpyraline hydrochloride (CHEBI:31508) has role H₁-receptor antagonist (CHEBI:37955) dithiadene (CHEBI:167625) has role H₁-receptor antagonist (CHEBI:37955) doxylamine (CHEBI:51380) has role H₁-receptor antagonist (CHEBI:37955) emedastine (CHEBI:4779) has role H₁-receptor antagonist (CHEBI:37955) emedastine difumarate (CHEBI:59865) has role H₁-receptor antagonist (CHEBI:37955) epinastine (CHEBI:51032) has role H₁-receptor antagonist (CHEBI:37955) fexofenadine (CHEBI:5050) has role H₁-receptor antagonist (CHEBI:37955) hydroxyzine (CHEBI:5818) has role H₁-receptor antagonist (CHEBI:37955) ketotifen (CHEBI:92511) has role H₁-receptor antagonist (CHEBI:37955) ketotifen fumarate (CHEBI:31750) has role H₁-receptor antagonist (CHEBI:37955) loratadine (CHEBI:6538) has role H₁-receptor antagonist (CHEBI:37955) mepyramine (CHEBI:6762) has role H₁-receptor antagonist (CHEBI:37955) methapyrilene (CHEBI:6820) has role H₁-receptor antagonist (CHEBI:37955) methapyrilene hydrochloride (CHEBI:38213) has role H₁-receptor antagonist (CHEBI:37955) mianserin (CHEBI:51137) has role H₁-receptor antagonist (CHEBI:37955) mirtazapine (CHEBI:6950) has role H₁-receptor antagonist (CHEBI:37955) orphenadrine (CHEBI:7789) has role H₁-receptor antagonist (CHEBI:37955) orphenadrine citrate (CHEBI:7790) has role H₁-receptor antagonist (CHEBI:37955) orphenadrine hydrochloride (CHEBI:60902) has role H₁-receptor antagonist (CHEBI:37955) oxatomide (CHEBI:31943) has role H₁-receptor antagonist (CHEBI:37955) paliperidone (CHEBI:82978) has role H₁-receptor antagonist (CHEBI:37955) paliperidone palmitate (CHEBI:83807) has role H₁-receptor antagonist (CHEBI:37955) pimozide (CHEBI:8212) has role H₁-receptor antagonist (CHEBI:37955) promazine (CHEBI:8459) has role H₁-receptor antagonist (CHEBI:37955) promethazine (CHEBI:8461) has role H₁-receptor antagonist (CHEBI:37955) promethazine hydrochloride (CHEBI:8462) has role H₁-receptor antagonist (CHEBI:37955) risperidone (CHEBI:8871) has role H₁-receptor antagonist (CHEBI:37955) sertindole (CHEBI:9122) has role H₁-receptor antagonist (CHEBI:37955) thioridazine (CHEBI:9566) has role H₁-receptor antagonist (CHEBI:37955) trazodone (CHEBI:9654) has role H₁-receptor antagonist (CHEBI:37955) trazodone hydrochloride (CHEBI:9655) has role H₁-receptor antagonist (CHEBI:37955) triprolidine (CHEBI:84116) has role H₁-receptor antagonist (CHEBI:37955) triprolidine hydrochloride (anh.) (CHEBI:84119) has role H₁-receptor antagonist (CHEBI:37955) triprolidine hydrochloride monohydrate (CHEBI:32265) has role H₁-receptor antagonist (CHEBI:37955) triprolidine(1+) (CHEBI:84117) has role H₁-receptor antagonist (CHEBI:37955) zuclopenthixol (CHEBI:51364) has role H₁-receptor antagonist (CHEBI:37955)

Synonyms	Sources
classical antihistamines	ChEBI
classical antihistaminics	ChEBI
H₁ antihistaminics	ChEBI
H₁ receptor antagonists	IUPHAR
H₁ receptor blockaders	ChEBI
H₁-receptor antagonists	ChEBI
H₁-receptor blocker	ChEBI
H₁-receptor blockers	ChEBI

Citation	Type	Source
22035879	PubMed citation	Europe PMC

Last Modified

29 October 2021