spacer
spacer

PDBsum entry 5tr6

Go to PDB code: 
Top Page protein ligands links
Transferase/transferase inhibitor PDB id
5tr6
Contents
Protein chain
272 a.a.
Ligands
7KG
EDO
Waters ×132

References listed in PDB file
Key reference
Title Discovery of tak-659 an orally available investigational inhibitor of spleen tyrosine kinase (syk).
Authors B.Lam, Y.Arikawa, J.Cramlett, Q.Dong, R.De jong, V.Feher, C.E.Grimshaw, P.J.Farrell, I.D.Hoffman, A.Jennings, B.Jones, J.Matuszkiewicz, J.Miura, H.Miyake, S.R.Natala, L.Shi, M.Takahashi, E.Taylor, C.Wyrick, J.Yano, J.Zalevsky, Z.Nie.
Ref. Bioorg Med Chem Lett, 2016, 26, 5947-5950. [DOI no: 10.1016/j.bmcl.2016.10.087]
PubMed id 27839918
Abstract
No abstract given.
PROCHECK
Go to PROCHECK summary
 Headers

 

spacer

spacer