 |
PDBsum entry 5hcx
|
|
|
|
 |
|
|
|
|
|
|
|
|
|
|
|
|
|
|
|
 |
|
|
|
 |
 |
 |
 |
 |
 |
 |
 |
 |
 |
 |
 |
 |
 |
 |
 |
 |
|
|
|
|
|
|
|
|
|
|
Transferase/transferase inhibitor
|
PDB id
|
|
|
|
5hcx
|
|
|
|
|
|
|
|
|
|
|
|
|
|
|
|
|
|
|
|
|
References listed in PDB file
|
 |
|
Key reference
|
 |
|
Title
|
 |
Discovery of a noncovalent, Mutant-Selective epidermal growth factor receptor inhibitor.
|
 |
|
Authors
|
 |
B.K.Chan,
E.J.Hanan,
K.K.Bowman,
M.C.Bryan,
D.Burdick,
E.Chan,
Y.Chen,
S.Clausen,
T.Dela vega,
J.Dotson,
C.Eigenbrot,
R.L.Elliott,
R.A.Heald,
P.S.Jackson,
J.D.Knight,
H.La,
M.D.Lainchbury,
S.Malek,
H.E.Purkey,
G.Schaefer,
S.Schmidt,
E.M.Seward,
S.Sideris,
L.Shao,
S.Wang,
S.K.Yeap,
I.Yen,
C.Yu,
T.P.Heffron.
|
 |
|
Ref.
|
 |
J Med Chem, 2016,
59,
9080-9093.
[DOI no: ]
|
 |
|
PubMed id
|
 |
|
 |
 |
|
Abstract
|
 |
|
No abstract given.
|
 |
|
|
|
|
 |