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PDBsum entry 5hcx

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Transferase/transferase inhibitor PDB id
5hcx
Contents
Protein chain
298 a.a.
Ligands
SO4
60B
Waters ×7

References listed in PDB file
Key reference
Title Discovery of a noncovalent, Mutant-Selective epidermal growth factor receptor inhibitor.
Authors B.K.Chan, E.J.Hanan, K.K.Bowman, M.C.Bryan, D.Burdick, E.Chan, Y.Chen, S.Clausen, T.Dela vega, J.Dotson, C.Eigenbrot, R.L.Elliott, R.A.Heald, P.S.Jackson, J.D.Knight, H.La, M.D.Lainchbury, S.Malek, H.E.Purkey, G.Schaefer, S.Schmidt, E.M.Seward, S.Sideris, L.Shao, S.Wang, S.K.Yeap, I.Yen, C.Yu, T.P.Heffron.
Ref. J Med Chem, 2016, 59, 9080-9093. [DOI no: 10.1021/acs.jmedchem.6b00995]
PubMed id 27564586
Abstract
No abstract given.
PROCHECK
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 Headers

 

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