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PDBsum entry 4r7i

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Transferase/transferase inhibitor PDB id
4r7i
Contents
Protein chain
290 a.a.
Ligands
STI
Waters ×55

References listed in PDB file
Key reference
Title Structure-Guided blockade of csf1r kinase in tenosynovial giant-Cell tumor.
Authors W.D.Tap, Z.A.Wainberg, S.P.Anthony, P.N.Ibrahim, C.Zhang, J.H.Healey, B.Chmielowski, A.P.Staddon, A.L.Cohn, G.I.Shapiro, V.L.Keedy, A.S.Singh, I.Puzanov, E.L.Kwak, A.J.Wagner, D.D.Von hoff, G.J.Weiss, R.K.Ramanathan, J.Zhang, G.Habets, Y.Zhang, E.A.Burton, G.Visor, L.Sanftner, P.Severson, H.Nguyen, M.J.Kim, A.Marimuthu, G.Tsang, R.Shellooe, C.Gee, B.L.West, P.Hirth, K.Nolop, M.Van de rijn, H.H.Hsu, C.Peterfy, P.S.Lin, S.Tong-Starksen, G.Bollag.
Ref. N Engl J Med, 2015, 373, 428-437. [DOI no: 10.1056/NEJMoa1411366]
PubMed id 26222558
Abstract
No abstract given.
PROCHECK
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 Headers

 

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