 |
PDBsum entry 4r7i
|
|
|
|
 |
|
|
|
|
|
|
|
|
|
|
|
|
|
|
|
 |
|
|
|
 |
 |
 |
 |
 |
 |
 |
 |
 |
 |
 |
 |
 |
 |
 |
 |
 |
|
|
|
|
|
|
|
|
|
|
Transferase/transferase inhibitor
|
PDB id
|
|
|
|
4r7i
|
|
|
|
|
|
|
|
|
|
|
|
|
|
|
|
|
|
|
|
|
References listed in PDB file
|
 |
|
Key reference
|
 |
|
Title
|
 |
Structure-Guided blockade of csf1r kinase in tenosynovial giant-Cell tumor.
|
 |
|
Authors
|
 |
W.D.Tap,
Z.A.Wainberg,
S.P.Anthony,
P.N.Ibrahim,
C.Zhang,
J.H.Healey,
B.Chmielowski,
A.P.Staddon,
A.L.Cohn,
G.I.Shapiro,
V.L.Keedy,
A.S.Singh,
I.Puzanov,
E.L.Kwak,
A.J.Wagner,
D.D.Von hoff,
G.J.Weiss,
R.K.Ramanathan,
J.Zhang,
G.Habets,
Y.Zhang,
E.A.Burton,
G.Visor,
L.Sanftner,
P.Severson,
H.Nguyen,
M.J.Kim,
A.Marimuthu,
G.Tsang,
R.Shellooe,
C.Gee,
B.L.West,
P.Hirth,
K.Nolop,
M.Van de rijn,
H.H.Hsu,
C.Peterfy,
P.S.Lin,
S.Tong-Starksen,
G.Bollag.
|
 |
|
Ref.
|
 |
N Engl J Med, 2015,
373,
428-437.
[DOI no: ]
|
 |
|
PubMed id
|
 |
|
 |
 |
|
Abstract
|
 |
|
No abstract given.
|
 |
|
|
|
|
 |