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PDBsum entry 4ejn
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Transferase/transferase inhibitor
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PDB id
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4ejn
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References listed in PDB file
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Key reference
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Title
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Discovery and optimization of a series of 3-(3-Phenyl-3h-Imidazo[4,5-B]pyridin-2-Yl)pyridin-2-Amines: orally bioavailable, Selective, And potent ATP-Independent akt inhibitors.
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Authors
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M.A.Ashwell,
J.M.Lapierre,
C.Brassard,
K.Bresciano,
C.Bull,
S.Cornell-Kennon,
S.Eathiraj,
D.S.France,
T.Hall,
J.Hill,
E.Kelleher,
S.Khanapurkar,
D.Kizer,
S.Koerner,
J.Link,
Y.Liu,
S.Makhija,
M.Moussa,
N.Namdev,
K.Nguyen,
R.Nicewonger,
R.Palma,
J.Szwaya,
M.Tandon,
U.Uppalapati,
D.Vensel,
L.P.Volak,
E.Volckova,
N.Westlund,
H.Wu,
R.Y.Yang,
T.C.Chan.
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Ref.
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J Med Chem, 2012,
55,
5291-5310.
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PubMed id
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Abstract
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No abstract given.
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