PDBsum entry 4aqc

Transferase

PDB id: 4aqc

Contents

Protein chain

291 a.a.

Ligands

88A ×2

SO4 ×5

Waters ×442

References listed in PDB file

Key reference

• Title: A selective, Orally bioavailable 1,2,4-Triazolo[1,5-A]pyridine-Based inhibitor of janus kinase 2 for use in anticancer therapy: discovery of cep-33779.
• Authors: B.J.Dugan, D.E.Gingrich, E.F.Mesaros, K.L.Milkiewicz, M.A.Curry, A.L.Zulli, P.Dobrzanski, C.Serdikoff, M.Jan, T.S.Angeles, M.S.Albom, J.L.Mason, L.D.Aimone, S.L.Meyer, Z.Huang, K.J.Wells-Knecht, M.A.Ator, B.A.Ruggeri, B.D.Dorsey.
• Ref.: J Med Chem, 2012, 55, 5243-5254.
• PubMed id: 22594690

Abstract

No abstract given.