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PDBsum entry 3oev
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Hydrolase/hydrolase inhibitor
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PDB id
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3oev
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Contents |
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250 a.a.
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235 a.a.
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241 a.a.
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242 a.a.
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233 a.a.
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237 a.a.
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243 a.a.
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222 a.a.
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204 a.a.
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198 a.a.
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212 a.a.
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222 a.a.
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233 a.a.
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196 a.a.
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References listed in PDB file
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Key reference
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Title
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Optimization of a series of dipeptides with a p3 threonine residue as non-Covalent inhibitors of the chymotrypsin-Like activity of the human 20s proteasome.
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Authors
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C.Blackburn,
C.Barrett,
J.L.Blank,
F.J.Bruzzese,
N.Bump,
L.R.Dick,
P.Fleming,
K.Garcia,
P.Hales,
Z.Hu,
M.Jones,
J.X.Liu,
D.S.Sappal,
M.D.Sintchak,
C.Tsu,
K.M.Gigstad.
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Ref.
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Bioorg Med Chem Lett, 2010,
20,
6581-6586.
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PubMed id
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Abstract
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No abstract given.
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