PDBsum entry 3mvl

Transferase

PDB id: 3mvl

Contents

Protein chain

339 a.a.

Ligands

38P ×2

Waters ×125

References listed in PDB file

Key reference

• Title: Discovery of 4-(5-(Cyclopropylcarbamoyl)-2-Methylphenylamino)-5-Methyl-N-Propylpyrrolo[1,2-F][1,2,4]triazine-6-Carboxamide (bms-582949), A clinical p38α map kinase inhibitor for the treatment of inflammatory diseases.
• Authors: C.Liu, J.Lin, S.T.Wrobleski, S.Lin, J.Hynes, H.Wu, A.J.Dyckman, T.Li, J.Wityak, K.M.Gillooly, S.Pitt, D.R.Shen, R.F.Zhang, K.W.Mcintyre, L.Salter-Cid, D.J.Shuster, H.Zhang, P.H.Marathe, A.M.Doweyko, J.S.Sack, S.E.Kiefer, K.F.Kish, J.A.Newitt, M.Mckinnon, J.H.Dodd, J.C.Barrish, G.L.Schieven, K.Leftheris.
• Ref.: J Med Chem, 2010, 53, 6629-6639.
• PubMed id: 20804198

Abstract

No abstract given.