PDBsum entry 2x8i

Transferase

PDB id: 2x8i

Contents

Protein chain

261 a.a.

Ligands

X8I

SO4 ×2

GOL

Waters ×241

References listed in PDB file

Key reference

• Title: Discovery of a novel class of triazolones as checkpoint kinase inhibitors--Hit to lead exploration.
• Authors: V.Oza, S.Ashwell, P.Brassil, J.Breed, C.Deng, J.Ezhuthachan, H.Haye, C.Horn, J.Janetka, P.Lyne, N.Newcombe, L.Otterbien, M.Pass, J.Read, S.Roswell, M.Su, D.Toader, D.Yu, Y.Yu, A.Valentine, P.Webborn, A.White, S.Zabludoff, X.Zheng.
• Ref.: Bioorg Med Chem Lett, 2010, 20, 5133-5138.
• PubMed id: 20673630

Abstract

No abstract given.