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References listed in PDB file
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Key references
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No key reference given in PDB file
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Secondary reference #1
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Title
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Crystal structures of two potent nonamidine inhibitors bound to factor xa.
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Authors
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M.Adler,
M.J.Kochanny,
B.Ye,
G.Rumennik,
D.R.Light,
S.Biancalana,
M.Whitlow.
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Ref.
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Biochemistry, 2002,
41,
15514-15523.
[DOI no: ]
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PubMed id
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Secondary reference #2
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Title
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Thiophene-Anthranilamides as highly potent and orally available factor xa inhibitors.
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Authors
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B.Ye,
D.O.Arnaiz,
Y.L.Chou,
B.D.Griedel,
R.Karanjawala,
W.Lee,
M.M.Morrissey,
K.L.Sacchi,
S.T.Sakata,
K.J.Shaw,
S.C.Wu,
Z.Zhao,
M.Adler,
S.Cheeseman,
W.P.Dole,
J.Ewing,
R.Fitch,
D.Lentz,
A.Liang,
D.Light,
J.Morser,
J.Post,
G.Rumennik,
B.Subramanyam,
M.E.Sullivan,
R.Vergona,
J.Walters,
Y.X.Wang,
K.A.White,
M.Whitlow,
M.J.Kochanny.
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Ref.
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J Med Chem, 2007,
50,
2967-2980.
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PubMed id
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Note In the PDB file this reference is
annotated as "TO BE PUBLISHED".
The citation details given above were identified by an automated
search of PubMed on title and author
names, giving a
percentage match of
93%.
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Secondary reference #3
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Title
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Substituted thiophene-Anthranilamides as potent inhibitors of human factor xa
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Authors
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B.Ye,
D.O.Arnaiz,
Y.-L.Chou,
B.D.Griedel,
R.Karanjawala,
W.Lee,
M.M.Morrissey,
K.L.Sacchi,
S.T.Sakata,
K.J.Shaw,
S.C.Wu,
Z.Zhao,
M.Adler,
S.Cheeseman,
W.P.Dole,
J.Ewing,
R.Fitch,
D.Lentz,
A.Liang,
D.Light,
J.Morser,
J.Post,
G.Rumennik,
B.Subramanyam,
M.E.Sullivan,
R.Vergona,
J.Walters,
Y.-X.Wang,
K.A.White,
M.Whitlow,
M.J.Kochanny.
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Ref.
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bioorg med chem, 2007,
15,
2127.
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PubMed id
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Secondary reference #4
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Title
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Structure-Activity relationships of substituted benzothiophene-Anthranilamide factor xa inhibitors.
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Authors
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Y.L.Chou,
D.D.Davey,
K.A.Eagen,
B.D.Griedel,
R.Karanjawala,
G.B.Phillips,
K.L.Sacchi,
K.J.Shaw,
S.C.Wu,
D.Lentz,
A.M.Liang,
L.Trinh,
M.M.Morrissey,
M.J.Kochanny.
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Ref.
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Bioorg Med Chem Lett, 2003,
13,
507-511.
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PubMed id
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Secondary reference #5
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Title
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Preparation, Characterization, And the crystal structure of the inhibitor zk-807834 (ci-1031) complexed with factor xa.
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Authors
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M.Adler,
D.D.Davey,
G.B.Phillips,
S.H.Kim,
J.Jancarik,
G.Rumennik,
D.R.Light,
M.Whitlow.
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Ref.
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Biochemistry, 2000,
39,
12534-12542.
[DOI no: ]
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PubMed id
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Secondary reference #6
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Title
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Crystal structures of human factor xa complexed with potent inhibitors.
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Authors
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S.Maignan,
J.P.Guilloteau,
S.Pouzieux,
Y.M.Choi-Sledeski,
M.R.Becker,
S.I.Klein,
W.R.Ewing,
H.W.Pauls,
A.P.Spada,
V.Mikol.
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Ref.
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J Med Chem, 2000,
43,
3226-3232.
[DOI no: ]
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PubMed id
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Secondary reference #7
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Title
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Discovery of n-[2-[5-[Amino(imino)methyl]-2-Hydroxyphenoxy]-3, 5-Difluoro-6-[3-(4, 5-Dihydro-1-Methyl-1h-Imidazol-2-Yl)phenoxy]pyridin-4-Yl]-N-Methylgl y cine (zk-807834): a potent, Selective, And orally active inhibitor of the blood coagulation enzyme factor xa.
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Authors
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G.B.Phillips,
B.O.Buckman,
D.D.Davey,
K.A.Eagen,
W.J.Guilford,
J.Hinchman,
E.Ho,
S.Koovakkat,
A.Liang,
D.R.Light,
R.Mohan,
H.P.Ng,
J.M.Post,
K.J.Shaw,
D.Smith,
B.Subramanyam,
M.E.Sullivan,
L.Trinh,
R.Vergona,
J.Walters,
K.White,
M.Whitlow,
S.Wu,
W.Xu,
M.M.Morrissey.
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Ref.
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J Med Chem, 1998,
41,
3557-3562.
[DOI no: ]
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PubMed id
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