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Hydrolase/hydrolase inhibitor
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PDB id
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1ewp
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Contents |
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* Residue conservation analysis
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PDB id:
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| Name: |
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Hydrolase/hydrolase inhibitor
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Title:
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Cruzain bound to mor-leu-hpq
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Structure:
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Cruzain. Chain: a. Fragment: catalytic domain. Synonym: cruzipain, cruzaine. Engineered: yes
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Source:
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Trypanosoma cruzi. Organism_taxid: 5693. Expressed in: escherichia coli. Expression_system_taxid: 562.
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Resolution:
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1.75Å
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R-factor:
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0.183
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R-free:
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0.206
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Authors:
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S.A.Gillmor
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Key ref:
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S.A.Gillmor
(1998).
Chapter 3: X-Ray structures of complexes of cruzain with designed covalent inhibitors.
Enzyme-Ligand interactions, Inhibition and specificity,
50-80.
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