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PDBe Entry: 4pax
THE CATALYTIC FRAGMENT OF POLY(ADP-RIBOSE) POLYMERASE COMPLEXED WITH 8-HYDROXY-2-METHYL-3-HYDRO-QUINAZOLIN-4-ONE
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| Summary | ![]() |
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| Header |
TRANSFERASE
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| Method | X-RAY DIFFRACTION | |||||||||||||
| Experiment | Resolution: 2.8 Å, R-factor: 16.7%, Spacegroup: P 21 21 21 | |||||||||||||
| Released | 27/05/1998, deposition: 25/11/1997, last revision: 24/02/2009 | |||||||||||||
| Authors |
Ruf, A. ; Schulz, G.E.
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| Primary citation |
Inhibitor and NAD+ binding to poly(ADP-ribose) polymerase as derived from crystal structures and homology modeling. BIOCHEMISTRY vol:37, pag:3893-3900 (1998) [PubMed ID 9521710 ]
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| Keywords |
TRANSFERASE , GLYCOSYLTRANSFERASE , NAD(+) ADP-RIBOSYLTRANSFERASE
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| EC |
2.4.2.30 ExPASy BRENDA (A)
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| Organism |
Gallus gallus(chicken) 9031 (A)
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| UniProt |
Poly [ADP-ribose] polymerase 1 (EC 2.4.2.30) (PARP-1) (ADPRT) (NAD(+) ADP-ribosyltransferase 1) (Poly[ADP-ribose] synthetase 1) P26446 (A)
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| Solvent | A | |||||||||||||
| Polymers |
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| Heterogens |
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