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PDBe Entry: 4pax view

THE CATALYTIC FRAGMENT OF POLY(ADP-RIBOSE) POLYMERASE COMPLEXED WITH 8-HYDROXY-2-METHYL-3-HYDRO-QUINAZOLIN-4-ONE
Summary
Header TRANSFERASEsearch
Method X-RAY DIFFRACTION
Experiment Resolution: 2.8 Å, R-factor: 16.7%, Spacegroup: P 21 21 21
Released 27/05/1998, deposition: 25/11/1997, last revision: 24/02/2009
Authors Ruf, A.search; Schulz, G.E.search
Primary citation Inhibitor and NAD+ binding to poly(ADP-ribose) polymerase as derived from crystal structures and homology modeling.
BIOCHEMISTRYsearch vol:37, pag:3893-3900 (1998) [PubMed ID 9521710 ]search
Keywords TRANSFERASEsearch, GLYCOSYLTRANSFERASEsearch, NAD(+) ADP-RIBOSYLTRANSFERASEsearch
EC 2.4.2.30 ExPASy BRENDA search (A)
Organism Gallus gallus(chicken) 9031search(A)
UniProt Poly [ADP-ribose] polymerase 1 (EC 2.4.2.30) (PARP-1) (ADPRT) (NAD(+) ADP-ribosyltransferase 1) (Poly[ADP-ribose] synthetase 1) P26446search (A)
Solvent A
Polymers
Id Name Type UniProt Residues Observed
A POLY(ADP-RIBOSE) POLYMERASE Protein P26446 (PARP1_CHICK)search
361 96%
Heterogens
Id Name Ligands
A 8-HYDROXY-2-METHYL-3-HYDRO-QUINAZOLIN-4-ONE NU1 search
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