Structure analysis

Crystal structure of the T315I Abl mutant in complex with the inhibitor PHA-739358

X-ray diffraction
2.5Å resolution
Source organism: Homo sapiens
Assembly composition:
monomeric (preferred)
Entry contents: 1 distinct polypeptide molecule

Assemblies

Assembly 1 (preferred)
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Multimeric state: monomeric
Accessible surface area: 13435.94 Å2
Buried surface area: 1035.71 Å2
Dissociation area: 468.92 Å2
Dissociation energy (ΔGdiss): -0.06 kcal/mol
Dissociation entropy (TΔSdiss): 5.4 kcal/mol
Symmetry number: 1
PDBe Complex ID: PDB-CPX-132602
Assembly 2
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Multimeric state: monomeric
Accessible surface area: 13481.56 Å2
Buried surface area: 1022.24 Å2
Dissociation area: 462.07 Å2
Dissociation energy (ΔGdiss): 0.57 kcal/mol
Dissociation entropy (TΔSdiss): 5.41 kcal/mol
Symmetry number: 1
PDBe Complex ID: PDB-CPX-132602

Macromolecules

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