Structure analysis

Androgen receptor LBD with small molecule

X-ray diffraction
2.1Å resolution
Source organism: Homo sapiens
Assembly composition:
monomeric (preferred)
Entry contents: 1 distinct polypeptide molecule

Assemblies

Assembly 1 (preferred)
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Multimeric state: monomeric
Accessible surface area: 12157.62 Å2
Buried surface area: 1134.33 Å2
Dissociation area: 341.52 Å2
Dissociation energy (ΔGdiss): -1.44 kcal/mol
Dissociation entropy (TΔSdiss): 3.8 kcal/mol
Symmetry number: 1
PDBe Complex ID: PDB-CPX-145222

Macromolecules

Chain: A
Length: 251 amino acids
Theoretical weight: 29.28 KDa
Source organism: Homo sapiens
Expression system: Escherichia coli
UniProt:
  • Canonical: P10275 (Residues: 670-920; Coverage: 27%)
Gene names: AR, DHTR, NR3C4
Pfam: Ligand-binding domain of nuclear hormone receptor
InterPro:
CATH: Retinoid X Receptor
SCOP: Nuclear receptor ligand-binding domain

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