Structure analysis

cFMS tyrosine kinase (tie2 KID) in complex with an arylamide inhibitor

X-ray diffraction
1.8Å resolution
Source organism: Homo sapiens
Assembly composition:
monomeric (preferred)
Entry contents: 1 distinct polypeptide molecule

Assemblies

Assembly 1 (preferred)
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Multimeric state: monomeric
Accessible surface area: 15260.36 Å2
Buried surface area: 769.88 Å2
Dissociation area: 384.94 Å2
Dissociation energy (ΔGdiss): -5.27 kcal/mol
Dissociation entropy (TΔSdiss): 4.44 kcal/mol
Symmetry number: 1
PDBe Complex ID: PDB-CPX-139513

Macromolecules

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