Structure analysis

EGFR kinase domain complexed with a quinazoline inhibitor- GW572016

X-ray diffraction
2.4Å resolution
Source organism: Homo sapiens
Assembly composition:
monomeric (preferred)
Entry contents: 1 distinct polypeptide molecule

Assemblies

Assembly 1 (preferred)
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Multimeric state: monomeric
Accessible surface area: 13378.26 Å2
Buried surface area: 1534.12 Å2
Dissociation area: 107.58 Å2
Dissociation energy (ΔGdiss): 5.94 kcal/mol
Dissociation entropy (TΔSdiss): 0.61 kcal/mol
Symmetry number: 1
PDBe Complex ID: PDB-CPX-132671

Macromolecules

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