Structure analysis

CRYSTAL STRUCTURE OF ESTROGEN RECEPTOR ALPHA COMPLEXED WITH WAY-244

X-ray diffraction
2.8Å resolution
Source organism: Homo sapiens
Assembly composition:
hetero tetramer (preferred)
Entry contents: 2 distinct polypeptide molecules

Assemblies

Assembly 1 (preferred)
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Multimeric state: hetero tetramer
Accessible surface area: 20436.37 Å2
Buried surface area: 6713.99 Å2
Dissociation area: 1,639.65 Å2
Dissociation energy (ΔGdiss): 6.8 kcal/mol
Dissociation entropy (TΔSdiss): 13.43 kcal/mol
Symmetry number: 2
PDBe Complex ID: PDB-CPX-136924

Macromolecules

Chains: A, B
Length: 245 amino acids
Theoretical weight: 28.06 KDa
Source organism: Homo sapiens
Expression system: Escherichia coli BL21(DE3)
UniProt:
  • Canonical: P03372 (Residues: 305-549; Coverage: 41%)
Gene names: ESR, ESR1, NR3A1
Pfam: Ligand-binding domain of nuclear hormone receptor
InterPro:
CATH: Retinoid X Receptor

Search similar proteins

Chains: C, D
Length: 13 amino acids
Theoretical weight: 1.58 KDa
Source organism: Homo sapiens
Expression system: Not provided

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