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PDBe Entry: 1i32 view

LEISHMANIA MEXICANA GLYCERALDEHYDE-3-PHOSPHATE DEHYDROGENASE IN COMPLEX WITH INHIBITORS
Summary
Header OXIDOREDUCTASEsearch
Method X-RAY DIFFRACTION
Experiment Resolution: 2.6 Å, R-factor: 20.5%, Free R-factor: 25.6%, Spacegroup: P 21 21 2
Released 03/10/2001, deposition: 12/02/2001, last revision: 24/02/2009
Authors Suresh, S.search; Bressi, J.C.search; Kennedy, K.J.search; Verlinde, C.L.M.J.search; Gelb, M.H.search; Hol, W.G.J.search
Primary citation Conformational changes in Leishmania mexicana glyceraldehyde-3-phosphate dehydrogenase induced by designed inhibitors.
J.MOL.BIOL.search vol:309, pag:423-435 (2001) [PubMed ID 11371162 ]search
Keywords enzymesearch, dehydrogenasesearch, OXIDOREDUCTASEsearch
EC 1.2.1.12 ExPASy BRENDA search (A B C D E F)
Organism Leishmania mexicana 5665search(A B C D E F)
UniProt Glyceraldehyde-3-phosphate dehydrogenase, glycosomal (EC 1.2.1.12) (GAPDH) Q27890search (A B C D E F)
Solvent A, B, C, D, E, F
Related entries 1gyp, 1gyq, 1i33
Polymers
Id Name Type UniProt Residues Observed
A, B, C, D, E, F GLYCERALDEHYDE 3-PHOSPHATE DEHYDROGENASE Protein Q27890 (G3PG_LEIME)search
360 99%
Heterogens
Id Name Ligands
A, B, C, D, E, F N-NAPHTHALEN-1-YLMETHYL-2'-[3,5-DIMETHOXYBENZAMIDO]-2'-DEOXY-ADENOSINE NMD search
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