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PDBe Entry: 1eed view

X-RAY CRYSTALLOGRAPHIC ANALYSIS OF INHIBITION OF ENDOTHIAPEPSIN BY CYCLOHEXYL RENIN INHIBITORS
Summary
Header ASPARTIC PROTEINASEsearch
Method X-RAY DIFFRACTION
Experiment Resolution: 2.0 Å, R-factor: 15.2%, Spacegroup: P 1 21 1
Released 31/01/1994, deposition: 15/06/1992, last revision: 25/08/2009
Authors Blundell, T.L.search; Frazao, C.search; Cooper, J.B.search
Primary citation X-ray crystallographic analysis of inhibition of endothiapepsin by cyclohexyl renin inhibitors.
BIOCHEMISTRYsearch vol:31, pag:8142-8150 (1992) [PubMed ID 1525155 ]search
Keywords ASPARTIC PROTEINASEsearch
EC 3.4.23.22 ExPASy BRENDA search (P)
Organism Cryphonectria parasitica 5116search(I)
UniProt Endothiapepsin precursor (EC 3.4.23.22) (Aspartate protease) P11838search (P)
Solvent I, P
Polymers
Id Name Type UniProt Residues Observed
I CYCLOHEXYL RENIN INHIBITOR PD125754 Mixed
4 100%
P ENDOTHIAPEPSIN Protein P11838 (CARP_CRYPA)search
330 100%
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